A Study Of Two Dual PI3K/mTOR Inhibitors, PF-04691502 And PF-05212384 In Patients With Recurrent Endometrial Cancer

This study is currently recruiting participants.
Verified June 2013 by Pfizer
Sponsor:
Information provided by (Responsible Party):
Pfizer
ClinicalTrials.gov Identifier:
NCT01420081
First received: August 17, 2011
Last updated: June 4, 2013
Last verified: June 2013
  Purpose

This study will investigate the individual safety and efficacy of two dual PI3K/mTOR inhibitors in patients with recurrent endometrial cancer.


Condition Intervention Phase
Endometrial Neoplasms
Drug: PF-05212384
Phase 2

Study Type: Interventional
Study Design: Allocation: Randomized
Endpoint Classification: Safety/Efficacy Study
Intervention Model: Parallel Assignment
Masking: Open Label
Primary Purpose: Treatment
Official Title: A Randomized Phase 2 Non-Comparative Study Of The Efficacy Of PF-04691502 And PF-05212384 In Patients With Recurrent Endometrial Cancer

Resource links provided by NLM:


Further study details as provided by Pfizer:

Primary Outcome Measures:
  • Number of Participants With Clinical Benefit Response (CBR) [ Time Frame: 16 ] [ Designated as safety issue: No ]

Secondary Outcome Measures:
  • Number of Participants With Objective Response [ Time Frame: 12 months ] [ Designated as safety issue: No ]
  • Overall Survival (OS) [ Time Frame: 12.0 ] [ Designated as safety issue: No ]
  • Progression-Free Survival (PFS) [ Time Frame: 12 ] [ Designated as safety issue: No ]
  • Progression-Free Survival (PFS) [ Time Frame: 6 ] [ Designated as safety issue: No ]
  • Area under the Concentration-Time Curve (AUC) [ Time Frame: Pre-dose, and post dose at 0.5, 1, 2, 3, 4, 6, and 24 hours post dose. Pre dose cycles 2, 3, 4 ] [ Designated as safety issue: No ]
  • Area under the Concentration-Time Curve (AUC) [ Time Frame: 0, 0.5, 1, 2, 4, 6, 24, 72, and 120 hours post dose and pre and 0.5 hour post dose cycles 2, 3, 4 ] [ Designated as safety issue: No ]
  • Expression and/or phosphorylation in biopsied tumor tissue of PI3K pathway proteins [ Time Frame: Baseline and 28 days ] [ Designated as safety issue: No ]
  • Gene and/or protein expression biomarkers in biopsied tumor tissue relating to PI3K and/or mTOR pathway activation [ Time Frame: Baseline ] [ Designated as safety issue: No ]

Estimated Enrollment: 144
Study Start Date: January 2012
Estimated Study Completion Date: May 2014
Estimated Primary Completion Date: May 2014 (Final data collection date for primary outcome measure)
Arms Assigned Interventions
Experimental: B
PI3K Basal, IV Compound
Drug: PF-05212384
154mg IV weekly
Other Name: PKI-587
Experimental: C
PI3K Activated, Oral Compound
Drug: PF-05212384
154mg IV weekly
Other Name: PKI-587
Experimental: F
Japanese lead in cohort, IV compound
Drug: PF-05212384
154mg IV weekly
Other Name: PKI-587

  Eligibility

Ages Eligible for Study:   20 Years and older
Genders Eligible for Study:   Female
Accepts Healthy Volunteers:   No
Criteria

Inclusion Criteria:

  • Recurrent endometrial carcinoma
  • Disease progression following one or two lines of prior treatment with platinum containing chemotherapy
  • Tumor tissue available at time of screening for PI3K analysis
  • Adequate performance status
  • Adequate glucose control, bone marrow, kidney, liver, and heart function

Exclusion Criteria:

  • More than 2 prior cytotoxic chemo regimens for endometrial carcinoma
  • Prior therapy with an agent known to be a PI3K, and or mTOR and or AKT inhibitor
  • Active brain metastases
  Contacts and Locations
Please refer to this study by its ClinicalTrials.gov identifier: NCT01420081

Contacts
Contact: Pfizer CT.gov Call Center 1-800-718-1021

  Hide Study Locations
Locations
United States, Alabama
Pfizer Investigational Site Recruiting
Birmingham, Alabama, United States, 35294
Pfizer Investigational Site Recruiting
Birmingham, Alabama, United States, 35249-7333
Pfizer Investigational Site Recruiting
Birmingham, Alabama, United States, 35249
Pfizer Investigational Site Recruiting
Birmingham, Alabama, United States, 35233
United States, California
Pfizer Investigational Site Recruiting
La Jolla, California, United States, 92093
Pfizer Investigational Site Recruiting
La Jolla, California, United States, 92037
Pfizer Investigational Site Recruiting
San Diego, California, United States, 92103
United States, Florida
Pfizer Investigational Site Recruiting
Coral Gables, Florida, United States, 33133
Pfizer Investigational Site Recruiting
Miami, Florida, United States, 33133
United States, Georgia
Pfizer Investigational Site Not yet recruiting
Augusta, Georgia, United States, 30912
United States, Illinois
Pfizer Investigational Site Recruiting
Chicago, Illinois, United States, 60637
United States, Kansas
Pfizer Investigational Site Not yet recruiting
Fairway, Kansas, United States, 66205
Pfizer Investigational Site Not yet recruiting
Kansas City, Kansas, United States, 66160
Pfizer Investigational Site Not yet recruiting
Westwood, Kansas, United States, 66205
United States, Louisiana
Pfizer Investigational Site Recruiting
Covington, Louisiana, United States, 70433
United States, Massachusetts
Pfizer Investigational Site Recruiting
Boston, Massachusetts, United States, 02215
Pfizer Investigational Site Recruiting
Boston, Massachusetts, United States, 02115
Pfizer Investigational Site Recruiting
Boston, Massachusetts, United States, 02114
United States, Michigan
Pfizer Investigational Site Not yet recruiting
Ann Arbor, Michigan, United States, 48109
United States, New Mexico
Pfizer Investigational Site Recruiting
Albuquerque, New Mexico, United States, 87106
United States, Pennsylvania
Pfizer Investigational Site Recruiting
Abington, Pennsylvania, United States, 19001
Australia, Victoria
Pfizer Investigational Site Recruiting
East Melbourne, Victoria, Australia, 3002
Canada, Alberta
Pfizer Investigational Site Not yet recruiting
Calgary, Alberta, Canada, T2N 4N2
Pfizer Investigational Site Not yet recruiting
Calgary, Alberta, Canada, T2N 2T9
Canada, British Columbia
Pfizer Investigational Site Recruiting
Vancouver, British Columbia, Canada, V5Z 4E6
Canada, Ontario
Pfizer Investigational Site Recruiting
Kingston, Ontario, Canada, K7L 5P9
Pfizer Investigational Site Recruiting
Toronto, Ontario, Canada, M5G 2M9
Canada, Quebec
Pfizer Investigational Site Not yet recruiting
Montreal, Quebec, Canada, H2L 4M1
Pfizer Investigational Site Recruiting
Montreal, Quebec, Canada, H3T 1E2
Japan
Pfizer Investigational Site Active, not recruiting
Nagoya, Aichi, Japan
Pfizer Investigational Site Active, not recruiting
Akashi, Hyogo, Japan
Pfizer Investigational Site Active, not recruiting
Hidaka, Saitama, Japan
Pfizer Investigational Site Active, not recruiting
Chuo-Ku, Tokyo, Japan
Poland
Pfizer Investigational Site Not yet recruiting
Lodz, Poland, 93-509
Pfizer Investigational Site Recruiting
Lublin, Poland, 20-090
Pfizer Investigational Site Not yet recruiting
Poznan, Poland, 61- 866
Pfizer Investigational Site Not yet recruiting
Poznan, Poland, 61-878
Russian Federation
Pfizer Investigational Site Recruiting
Krasnodar, Russian Federation, 350040
Pfizer Investigational Site Recruiting
Pyatigorsk, Russian Federation, 35702
Pfizer Investigational Site Not yet recruiting
Ryazan, Russian Federation, 390011
Pfizer Investigational Site Recruiting
Saint Petersburg, Russian Federation, 198255
Pfizer Investigational Site Not yet recruiting
Ufa, Russian Federation, 450054
Slovakia
Pfizer Investigational Site Not yet recruiting
Bratislava, Slovakia, 833 10
Pfizer Investigational Site Not yet recruiting
Presov, Slovakia, 08001
Spain
Pfizer Investigational Site Recruiting
Barcelona, Spain, 08035
Pfizer Investigational Site Not yet recruiting
Madrid, Spain, 28046
Pfizer Investigational Site Recruiting
Madrid, Spain, 28033
Pfizer Investigational Site Recruiting
Madrid, Spain, 28040
Pfizer Investigational Site Recruiting
Valencia, Spain, 46009
United Kingdom
Pfizer Investigational Site Recruiting
London, England, United Kingdom, SW3 6JJ
Pfizer Investigational Site Not yet recruiting
Glasgow, Scotland, United Kingdom
Pfizer Investigational Site Not yet recruiting
Bebington, Wirral, United Kingdom, CH63 4JY
Pfizer Investigational Site Not yet recruiting
London, United Kingdom, NW1 2PG
Sponsors and Collaborators
Pfizer
Investigators
Study Director: Pfizer CT.gov Call Center Pfizer
  More Information

Additional Information:
No publications provided

Responsible Party: Pfizer
ClinicalTrials.gov Identifier: NCT01420081     History of Changes
Other Study ID Numbers: B1271004
Study First Received: August 17, 2011
Last Updated: June 4, 2013
Health Authority: United States: Food and Drug Administration

Keywords provided by Pfizer:
uterine neoplasms
endometrial
uterine
cancer
PI3K
mTOR
PI3K/mTOR
recurrent
metastatic

Additional relevant MeSH terms:
Neoplasms
Endometrial Neoplasms
Adenoma
Uterine Neoplasms
Genital Neoplasms, Female
Urogenital Neoplasms
Neoplasms by Site
Uterine Diseases
Genital Diseases, Female
Neoplasms, Glandular and Epithelial
Neoplasms by Histologic Type

ClinicalTrials.gov processed this record on June 18, 2013