Effect of Spinal Ketorolac After Acute Opioid Exposure

This study is ongoing, but not recruiting participants.
Sponsor:
Collaborator:
Information provided by (Responsible Party):
James C. Eisenach, M.D., Wake Forest University
ClinicalTrials.gov Identifier:
NCT00693160
First received: February 15, 2008
Last updated: February 14, 2012
Last verified: February 2012
  Purpose

This research study is being done because pain is a significant problem for patients with a variety of medical problems and following surgery or traumatic injury. Currently available pain medications may not treat all types of pain or may treat pain only at doses that produce side effects and complications. The medication in this study may have a role in better treatment of pain. The goals of this study are to see if a dose of ketorolac (non-narcotic, pain reliever), given into the fluid in your back near the spine has any effect on pain or discomfort in the skin sensation that will take place after applying capsaicin (chili pepper) cream. The sunburn-like sensation that people experience after having capsaicin cream applied is similar to, but much milder than, the pain that some people have after surgery and after certain types of nerve injuries. This study will test the effects of combining two medications that are often given together to control postoperative pain or pain from a nerve injury. The investigators are especially interested in answering two questions about the effects of ketorolac (non-narcotic pain reliever) and remifentanil (intravenous [IV] narcotic painkiller):

  1. How much does remifentanil (narcotic painkiller) affect the sunburn-like painful area on your skin, which develops after applying capsaicin cream?
  2. What pain relieving effects does spinal ketorolac have when given with IV remifentanil?

Condition Intervention Phase
Healthy
Drug: ketorolac
Drug: placebo
Drug: remifentanil
Phase 2

Study Type: Interventional
Study Design: Allocation: Randomized
Endpoint Classification: Efficacy Study
Intervention Model: Parallel Assignment
Masking: Double Blind (Subject, Investigator, Outcomes Assessor)
Primary Purpose: Basic Science
Official Title: Effect of Intrathecal Ketorolac on Mechanical Hypersensitivity Following Acute Opioid Exposure

Resource links provided by NLM:


Further study details as provided by Wake Forest University:

Primary Outcome Measures:
  • primary outcome measure is the area of hyperalgesia [ Time Frame: 24 hours ] [ Designated as safety issue: No ]

Secondary Outcome Measures:
  • secondary outcome measure is the CSF PGE2 concentration after stopping remifentanil [ Time Frame: 2.5 hours ] [ Designated as safety issue: No ]

Estimated Enrollment: 50
Study Start Date: December 2007
Estimated Study Completion Date: August 2012
Estimated Primary Completion Date: August 2012 (Final data collection date for primary outcome measure)
Arms Assigned Interventions
Active Comparator: 1
subject will receive a single intrathecal injection of ketorolac 2 mg
Drug: ketorolac
single intrathecal injection of ketorolac 2 mg
Other Names:
  • ketorolac
  • toradol
  • acular pf
Drug: remifentanil
All subjects will receive a remifentanil infusion
Other Name: ultiva
Placebo Comparator: 2
subject will receive a single intrathecal injection of placebo (preservative-free normal saline)
Drug: placebo
subject will receive a placebo (preservative free normal saline) spinal injection
Other Name: placebo
Drug: remifentanil
All subjects will receive a remifentanil infusion
Other Name: ultiva

Detailed Description:

Intravenous (IV) remifentanil stimulates spinal COX activity, leading to increased CSF PGE2 concentrations and areas of capsaicin-induced mechanical hypersensitivity after remifentanil infusion, and these effects will be blocked by intrathecal ketorolac.

Areas of mechanical hyperalgesia and allodynia will be established by topical capsaicin + intermittent heat in healthy volunteers, who will be randomized to receive intrathecal saline or ketorolac during remifentanil infusion, with primary outcome measure area of hyperalgesia and secondary outcome measure CSF PGE2 concentration after stopping remifentanil.

  Eligibility

Ages Eligible for Study:   18 Years to 55 Years
Genders Eligible for Study:   Both
Accepts Healthy Volunteers:   Yes
Criteria

Inclusion Criteria:

  • healthy
  • ASA I or II classification
  • between the ages of 18-55
  • weigh less than 250 pounds
  • without chronic pain

Exclusion Criteria:

  • taking analgesics in the last 2 weeks
  • positive urine drug screen
  • pregnancy
  • currently taking any prescription antidepressants or other medications that are mood altering
  • liver or kidney disease
  • stomach ulcers
  • allergies to ketorolac, lidocaine, or capsaicin cream
  • lung disease (COPD)
  Contacts and Locations
Please refer to this study by its ClinicalTrials.gov identifier: NCT00693160

Locations
United States, North Carolina
Wake Forest University Health Sciences
Winston-Salem, North Carolina, United States, 27157
Sponsors and Collaborators
Wake Forest University
Investigators
Principal Investigator: James C. Eisenach, M.D. Wake Forest University
  More Information

No publications provided

Responsible Party: James C. Eisenach, M.D., Professor, Wake Forest University
ClinicalTrials.gov Identifier: NCT00693160     History of Changes
Other Study ID Numbers: IRB00002457, GM48085
Study First Received: February 15, 2008
Last Updated: February 14, 2012
Health Authority: United States: Food and Drug Administration

Keywords provided by Wake Forest University:
healthy volunteers
analgesia
pain
Healthy subjects

Additional relevant MeSH terms:
Ketorolac
Ketorolac Tromethamine
Remifentanil
Analgesics, Opioid
Anti-Inflammatory Agents, Non-Steroidal
Analgesics, Non-Narcotic
Analgesics
Sensory System Agents
Peripheral Nervous System Agents
Physiological Effects of Drugs
Pharmacologic Actions
Anti-Inflammatory Agents
Therapeutic Uses
Antirheumatic Agents
Cyclooxygenase Inhibitors
Enzyme Inhibitors
Molecular Mechanisms of Pharmacological Action
Central Nervous System Agents
Central Nervous System Depressants
Hypnotics and Sedatives
Anesthetics, Intravenous
Anesthetics, General
Anesthetics

ClinicalTrials.gov processed this record on May 16, 2013